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9781493914005: Discovering and Developing Molecules with Optimal Drug-Like Properties

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Sinopsis

.- 1 Developability Assessment and Risk Management During Drug Discovery

 

.- 2 Discovery Formulations - Approaches and Practices in Early Preclinical Development

 

.- 3 Enabling Discovery Through Leveraging and Miniaturizing Pharmaceutical Principles and Processes

 

.- 4 Diagnosing Biopharmaceutical Limitations

 

.- 5 The Importance of Molecular Design Principles in Delivering High Quality Pharmaceutical Candidates

 

.- 6 Predictive Approaches to Establishing, Understanding, and Communicating Risk with Emphasis on Early Development

 

.- 7 Strategies and Methods for Drug Candidate Phase Optimization in Discovery Space

.- 8 Efficient Laboratory Methods to Assess Risk and Design Formulations

 

.- 9 Advanced X-ray Analytical Methods to Understand Structure, Properties and Risk

 

.- 10 Performance and Characterization of Amorphous Solid Dispersions: An Overview

 

.- 11 Hot-Melt Extrusion: The Process-Product-Performance Interplay

 

.- 12 Practical Considerations for Spray Dried Formulation and Process Development

 

.- 13 Nanosizing: "End-to-End" Formulation Strategy for Poorly-Water- Soluble Molecules

 

.- 14 Leveraging Solid State Form and Physiochemical Properties for Early Clinical Formulation Efforts:   Opportunities and Challenges during Telcagepant Liquid Capsule Development.

"Sinopsis" puede pertenecer a otra edición de este libro.

Otras ediciones populares con el mismo título

9781493913985: Discovering and Developing Molecules with Optimal Drug-Like Properties: 15 (AAPS Advances in the Pharmaceutical Sciences Series)

Edición Destacada

ISBN 10:  1493913980 ISBN 13:  9781493913985
Editorial: Springer, 2014
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